Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1046 |
Mexiletine hydrochloride
KOE-1173 (hydrochloride),Mexiletine HCl,KO1173,盐酸美西律 |
AhR; Sodium Channel | Immunology/Inflammation; Membrane transporter/Ion channel; Metabolism |
Mexiletine hydrochloride (KOE-1173 hydrochloride) 是一种电压门控钠通道阻滞剂,是 IB 类抗心律失常药。 Mexiletine hydrochloride 通过抑制心肌细胞内钠电流,从而降低心脏动作电位(0相)上升速率,并且降低浦肯野纤维的自律性而发挥抗心律失常作用。 | |||
T12023 |
Mexiletine-d6 hydrochloride
KOE-1173 D6 hydrochloride,Mexiletine D6 hydrochloride |
Others | Others |
Mexiletine D6 hydrochloride is a non-selective voltage-gated sodium channel blocker,is a Class IB antianhythmic. |